Diferencia entre revisiones de «Ivermectin»

 
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==General==
==General==
*Type: antiparasitic
*Type: [[antiparasitic]]
*Dosage Forms: 3
*Dosage Forms: Tablet, 3mg
*Common Trade Names: Stromectol
*Common Trade Names: Stromectol


==Adult Dosing==
==Adult Dosing==
'''[[strongyloidiasis]]''': 0.2 mg/kg PO x1
===[[Strongyloidiasis]]===
*0.2mg/kg PO x1


'''[[onchocerciasis]]''': 0.15 mg/kg PO x1
===[[Onchocerciasis]]===
*0.15mg/kg PO x1


'''[[scabies]], non-crusted''': 0.2 mg/kg PO x1
===[[Scabies]], non-crusted===
*0.2mg/kg PO x1


'''[[scabies]], crusted''': 0.2 mg/kg PO x1 on days 1,2,8,9,15
===[[Scabies]], crusted===
*0.2mg/kg PO x1 on days 1,2,8,9,15


'''[[pediculosis capitis]]''': 0.2 mg/kg pO q10 days x2 doses
===[[Pediculosis capitis]]===
*0.2mg/kg pO q10 days x2 doses


'''[[pediculosis corporis]]''': 12 mg PO q7 days x3 doses
===[[Pediculosis corporis]]===
*12mg PO q7 days x3 doses


'''[[pediculosis pubis]]''': 0.25 mg/kg PO q2wk x2 doses
===[[Pediculosis pubis]]===
*0.25mg/kg PO q2wk x2 doses


==Pediatric Dosing==
==Pediatric Dosing==
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==See Also==
==See Also==


==Sources==


==References==
<references/>
<references/>
[[Category:Drugs]]
 
[[Category:Pharmacology]]
[[Category:ID]]

Revisión actual - 20:51 22 sep 2019

General

  • Type: antiparasitic
  • Dosage Forms: Tablet, 3mg
  • Common Trade Names: Stromectol

Adult Dosing

Strongyloidiasis

  • 0.2mg/kg PO x1

Onchocerciasis

  • 0.15mg/kg PO x1

Scabies, non-crusted

  • 0.2mg/kg PO x1

Scabies, crusted

  • 0.2mg/kg PO x1 on days 1,2,8,9,15

Pediculosis capitis

  • 0.2mg/kg pO q10 days x2 doses

Pediculosis corporis

  • 12mg PO q7 days x3 doses

Pediculosis pubis

  • 0.25mg/kg PO q2wk x2 doses

Pediatric Dosing

Special Populations

  • Pregnancy Rating: C
  • Lactation: Safety Unknown
  • Renal Dosing- not defined
  • Hepatic Dosing- not defined

Contraindications

  • Allergy to class/drug

Adverse Reactions

Serious

Common

  • pruritus
  • rash
  • fever
  • edema
  • lymphadenopathy
  • headache
  • myalgia
  • dizziness
  • tachycardia
  • abnormal eye sensation
  • limbitis
  • conjunctivitis
  • ocular inflammation
  • hypotension, orthostatic
  • ALT, AST elevated
  • eosinophilia

Pharmacology

  • Half-life: 18h
  • Metabolism: liver, CYP450: unknown
  • Excretion: feces primarily, urine < 1%
  • Mechanism of Action: increases invertebrate nerve and muscle cell membrane permeability by binding to chloride ion channels, resulting in paralysis and death of parasite

See Also

References