Diferencia entre revisiones de «Alpha blockers»

(Text replacement - "Alpha" to "α")
Sin resumen de edición
 
(No se muestran 5 ediciones intermedias de 3 usuarios)
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==Background==
==Background==
*Also known as α-blockers
*Also known as α-blockers
**&α;<sub>1</sub>-blockers act on &α;<sub>1</sub>-adrenoceptors
**α<sub>1</sub>-blockers act on α<sub>1</sub>-adrenoceptors
**&α;<sub>2</sub>-blockers act on &α;<sub>2</sub>-adrenoceptors
**α<sub>2</sub>-blockers act on α<sub>2</sub>-adrenoceptors
*Act as neutral antagonists or inverse agonists of &α;-adrenergic receptors (α-adrenoceptors)
*Act as neutral antagonists or inverse agonists of α-adrenergic receptors (α-adrenoceptors)


==Medications==
==Medications==
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*Typical and atypical [[antipsychotics]]
*Typical and atypical [[antipsychotics]]


===Selective α 1===
===Selective α<sub>1</sub>===
*[[Alfuzosin]]
*[[Alfuzosin]]
*[[Doxazosin]]
*[[Doxazosin]]
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*[[Silodosin]]
*[[Silodosin]]


===Selective α 2===
===Selective α<sub>2</sub>===
*[[Atipamezole]]
*[[Atipamezole]]
*[[Idazoxan]]
*[[Idazoxan]]
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===Mixed===
===Mixed===
*The agents [[carvedilol]] and [[labetalol]] are both α- and [[beta blocker|&beta;-blockers]].
*The agents [[carvedilol]] and [[labetalol]] are both α- and [[β-blocker|&beta;-blockers]].


==Uses==
==Uses==
*[[hypertension]]
*[[hypertension]]
*[[Raynaud's disease]]
*[[Raynaud’s disease]]
*[[scleroderma]]
*[[scleroderma]]
*[[generalized anxiety disorder]]
*[[generalized anxiety disorder]]
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*[[Antihypertensive medications]]
*[[Antihypertensive medications]]
*[[Beta blocker]]
*[[Beta blocker]]
*[[Yohimbine toxicity]]


==References==
==References==
<references/>
<references/>
[[Category:Pharmacology]]
[[Category:Pharmacology]]

Revisión actual - 14:28 19 oct 2019

Background

  • Also known as α-blockers
    • α1-blockers act on α1-adrenoceptors
    • α2-blockers act on α2-adrenoceptors
  • Act as neutral antagonists or inverse agonists of α-adrenergic receptors (α-adrenoceptors)

Medications

Non-selective

Selective α1

Selective α2

Mixed

Uses

See also

References